Palladium-catalyzed conjugate addition of arylsulfonyl hydrazides to α,β-unsaturated ketones.

نویسندگان

  • Wen Chen
  • Hui Chen
  • Fuhong Xiao
  • Guo-Jun Deng
چکیده

A palladium-catalyzed desulfitative-denitrogenative conjugate addition of arylsulfonyl hydrazides to α,β-unsaturated ketones is described. The reaction showed very good selectivity and tolerated a wide range of functionalities under an atmosphere of oxygen with or without the aid of a metal co-oxidant.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 11 26  شماره 

صفحات  -

تاریخ انتشار 2013